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Pharmaceuticals/Chemicals

Aromasin (Exemestane)

Exemestane · Exe · Suicidal AI

Steroidal (suicidal) aromatase inhibitor; permanently inactivates aromatase enzyme.

Pharmacokinetic summary

Model tier
Advanced (t½ + Cmax + Tmax + F)
Half-life
0.9 days
Cmax
57.6 ng/mL
Tmax
0.1 days
Bioavailability
5%
Typical dose
6.25–25 mg