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Pharmaceuticals/Chemicals

Arimidex (Anastrozole)

Anastrozole · Adex · AI

Non-steroidal aromatase inhibitor; used to control estradiol on-cycle. Over-suppression risk.

Pharmacokinetic summary

Model tier
Advanced (t½ + Cmax + Tmax + F)
Half-life
2 days
Cmax
3930 ng/mL
Tmax
0.0 days
Bioavailability
80%
Typical dose
0.25–1 mg